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Cas No. |
Product name |
1116235-97-2 |
GSK1838705A |
more... |
GSK1838705A is a potent IGF-1R inhibitor with IC50 of 2.0 nM, modestly potent to IR and ALK with IC50 of 1.6 nM and 0.5 nM, respectively, and little activity to other protein... |
475488-23-4 |
NVP-ADW742 |
more... |
NVP-ADW742(ADW742; GSK 552602A ) is an selective IGF-1R inhibitor with IC50 of 0.17 μM, >16-fold more potent against IGF-1R than InsR; little activity to HER2, PDGFR, VEGF... |
196868-63-0 |
PQ401 |
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PQ401, a selective insulin-like growth factor-1 receptor blocker, is a novel diarylurea compound that inhibits IGF1R autophosphorylation with IC50 < 1 uM. |
1454846-35-5 |
PF-06463922 |
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PF-06463922 is a potent, dual ALK/ROS1 inhibitor with Ki of <0.02 nM, <0.07 nM, and 0.7 nM for ROS1, ALK (WT), and ALK (L1196M), respectively. Phase 1. |
1108743-60-7 |
Entrectinib |
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Entrectinib(NMS-E628、RXDX-101) is an orally available ALK inhibitor; exhibits good activity against NPM–ALK with an IC50 value of 55 nM. |
1022958-60-6 |
CEP28122 |
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CEP-28122 is a highly potent and selective orally active ALK inhibitor with IC50 of 1.9 ± 0.5 nM in an enzyme-based TRF assay. |
1391712-60-9 |
CEP-37440 |
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CEP-37440 is a novel potent and selective Dual FAK/ALK inhibitor with IC50 s of 2.3 nM (FAK) and 120 nM(ALK cellular IC50 in 75% human plasma). |
1627503-67-6 |
LDN-214117 |
more... |
LDN-214117 is a potent and selective BMP type I receptor kinase ALK2 inhibitor with IC50 of 24 nM. |
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